Peptide Active Data Details
Basic Peptide Information
DICL ID
DICL_Pep_04689
Ion Channel
Potassium channel subfamily K member 3
Peptide Function
Inhibitor
Gene Name
KCNK3
Activity Data (nM)
IC50
Not available
Ki
Not available
EC50
10 nM
Kd
Not available
Biologically Active
Not specified
Sequence Information
Peptide Sequence
CSCSSLMDKECVYFCHLDIIW
Peptide UniProt Accession
Not available
UniParc
UPI000002E63D
Peptide Synonyms/Alias
[Endothelin-1; ET-1; Endothelin I; 123626-67-5; CHEMBL3775234; 1-(4-Hydroxyphenyl)-2;4;6-triphenylpyridinium hydroxide inner salt hydrate; GTPL989; BDBM50155246; Endothelin 1; >=97.0% (HPLC); Endothelin 1; >=97% (HPLC); powder; Endothelin 1??; Vetec(TM) reagent grade; >=97%; L-cysteinyl-L-seryl-L-cysteinyl-L-seryl-L-seryl-L-leucyl-L-methionyl-L-alpha-aspartyl-L-lysyl-L-alpha-glutamyl-L-cysteinyl-L-valyl-L-tyrosyl-L-phenylalanyl-L-cysteinyl-L-histidyl-L-leucyl-L-alpha-aspartyl-L-isoleucyl-L-isoleucyl-L-tryptophan (1->15);(3->11)-bis(disulfide)]
Peptide Species
Not specified
Peptide Name
Not available
CAS Number
123626-67-5
Experimental Conditions
pH
pH 7.4
Holding Potential (mV)
−100 to 50 mV
Temperature
Not mention
Test Method
Patch-clamping
Test Species
CHO cell (Chinese hamster ovary cell)
Binding Information
Binding Site
Not specified
Binding Site Residue
Not specified
Ion Channel Information
Gene Abbreviation (ABB)
K2P
Ion Channel UniProt Accession
Source Organism
Homo sapiens (Human)
References & Disease Information
Disease
Not specified
PubChem CID
URL
Not available
PMID
Patent
Not available